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Ngwakọta kemịkalụ Sitagliptin Phosphate

Ngwakọta kemịkalụ Sitagliptin Phosphate

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Sitagliptin phosphate bụ dipeptidyl peptidase Ⅳ (DDP-4) klaasị inhibitor ọgwụ nke German Merck ụlọ ọrụ mepụtara ma buru ụzọ nweta nkwado US Food and Drug Administration maka ọgwụgwọ ụdị ọrịa shuga 2, bụ ọgwụ antidiabetic ọhụrụ, nwere ike imeziwanye ahụ nke ya. ike ibelata ọkwa glucose ọbara dị elu, yana mmụba dịtụ na-abawanye site na igbochi ọrụ nke enzyme a, gụnyere ọkwa glucagon-dị ka peptide 1 na insulinotropic peptide na-adabere na glucose, si otú ahụ na-akpali pancreas iji meziwanye mmepụta insulin ma kwụsị glucose. mmepụta na imeju, na n'ikpeazụ belata mmetụta ụlọ ọgwụ nke mkpokọta glucose ọbara.

  • Ọdịdị:ọcha siri ike
  • Nyocha:≥99.0%
  • Ebe mgbari:274.3 ℃
  • Ebe esi mmiri:529.9 ℃
  • Ebe mgbaze:202-204 ℃
  • Nkọwa ngwaahịa

    Mkpado ngwaahịa

    Nkọwa ngwaahịa

    Aha ngwaahịa Sitagliptin Phosphate CAS NO654671-78-0
    Ụdị okwu   (3R) -3-Amino-1-[3- (trifluoromethyl) -5,6-dihydro [1,2,4] triazolo [4,3-a] pyrazin-7 (8H) -yl] -4-( 2,4,5-trifluorophenyl) -1-butanone phosphate (1: 1);
    1-Butanone, 3-amino-1-[5,6-dihydro-3- (trifluoromethyl) -1,2,4-triazolo [4,3-a] pyrazin-7 (8H) -yl] -4- ( 2,4,5-trifluorophenyl) -, (3R) -, phosphate (1: 1);
    (3R) -3-amino-1-[3- (trifluoromethyl) -5,6-dihydro [1,2,4] triazolo [4,3-a] pyrazin-7 (8H) -yl] -4-( 2,4,5-trifluorophenyl) butan-1-otu phosphate (1: 1);
    CAS NO 654671-78-0
    Usoro ihe omimi C16H18F6N5O5P
    Ibu molekụla 505.31
    EINECS NO 1806241-263-5
    MDL NO MFCD22628883

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